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Cat. No. Product Name Target Signaling Pathways
T3120 K858 (Racemic)

K858 Racemic,K858

Apoptosis; Kinesin Apoptosis; Cytoskeletal Signaling
K858 Racemic (K858) 是一种选择性有丝分裂驱动蛋白 Eg5 抑制剂,以 ATP 非竞争性方式起作用,IC50值为 1.3 μM。
T12351 p53 and MDM2 proteins-interaction-inhibitor (racemic)

p53-and-mdm2-proteins-interaction-inhibitor-racemic

Others Others
p53 and MDM2 proteins-interaction-inhibitor (racemic) is an inhibitor of the interaction between p53 and MDM2 proteins.
T22253 AG-120 (racemic)

1-(4-氰基-2-吡啶基)-5-氧代-L-脯氨酰-2-(2-氯苯基)-N-(3,3-二氟环丁基)-N2-(5-氟-3-吡啶基)甘氨酰胺

Dehydrogenase Metabolism
AG-120 (racemic) 是 AG-120 的外消旋混合物,是一种可口服的异柠檬酸脱氢酶 1 型 (IDH1) 抑制剂,具有潜在的抗肿瘤活性。

化合物

K858 (Racemic)
Cat.No: T3120
Synonym: K858 Racemic,K858
Target: Apoptosis, Kinesin
p53 and MDM2 proteins-interaction-inhibitor (racemic)
Cat.No: T12351
Synonym: p53-and-mdm2-proteins-interaction-inhibitor-racemic
Target: Others
AG-120 (racemic)
Cat.No: T22253
Synonym: 1-(4-氰基-2-吡啶基)-5-氧代-L-脯氨酰-2-(2-氯苯基)-N-(3,3-二氟环丁基)-N2-(5-氟-3-吡啶基)甘氨酰胺
Target: Dehydrogenase
TargetMol Loading
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